• 专利附录
  • 专利说明
  • 权利要求
  • 类似技术
  • 同族专利
  • 引用文献
  • 法律状态
  • 优先权
    • 专利摘要:
    The method of obtaining piperidine derivatives of the general formula CO- (N -l, N 1 H 2 R 2 where R and R j are the same or different and mean hydrogen, alkyl with 1-4 carbon atoms, benzyl or together a group. - (cf) or their acid additive with s, characterized in that the compound of the general formula CHjO vx fN NH2 S where X is chlorine, bromine or alkylthio with 1-4 carbon atoms, is reacted with the compound of the general formula - C where R and Rj have the indicated meanings, followed by allocation of the target product in free form or as an acid addition salt.
    公开号:SU1187720A3
    申请号:SU833641410
    申请日:1983-09-13
    公开日:1985-10-23
    发明作者:Ментруп Антон；Рент Эрнст-Отто；Шромм Курт；Хефке Вольфганг；Гаида Вольфрам
    申请人:Берингер Ингельгейм Кг (Фирма)；
    IPC主号:
    专利说明:

    Table 1
    SN323
    CH,
    H
    sn.
    CH,
    CjHj135
    four
    80
    H
    - (CHj) -140
    6C.HS
    . H-CjH,
    H
    CjHj-CHjH
    92
    90
    88
    89.5
    91.5
    90
    92.5
    89
    权利要求:
    Claims (1)
    [1]
    A method of obtaining piperidine derivatives of the general formula nh 2 or alkylthio with the number of carbon atoms 1-4, is subjected to interaction with the compound of the general formula n / у ^ С0 “
    4 CO-CR t * 2 where R and R 2 have the indicated meanings, followed by the inclusion of the target product in free form or in the form of an acid addition salt.
    where X is chlorine, bromine
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    同族专利:
    公开号 | 公开日
    AU1939683A|1984-03-29|
    NO833423L|1984-03-26|
    ES8504181A1|1985-04-01|
    JPS5978187A|1984-05-04|
    PL243878A1|1985-01-02|
    PH20015A|1986-08-28|
    ES8504182A1|1985-04-01|
    US4539323A|1985-09-03|
    NZ205716A|1985-08-30|
    DD212517A5|1984-08-15|
    DK436583A|1984-03-26|
    CS235342B2|1985-05-15|
    FI833292A0|1983-09-15|
    DE3235565A1|1984-03-29|
    ES534351A0|1985-04-01|
    ZA837081B|1985-05-29|
    GR78973B|1984-10-02|
    DK436583D0|1983-09-23|
    HU191637B|1987-03-30|
    ES8501762A1|1984-12-01|
    AU561118B2|1987-04-30|
    PL139590B1|1987-02-28|
    IL69777A|1986-09-30|
    ES534349A0|1985-04-01|
    ES534350A0|1985-04-01|
    CA1215981A|1986-12-30|
    EP0104445A3|1985-07-10|
    FI833292A|1984-03-26|
    ES8504180A1|1985-04-01|
    PT77380A|1983-10-01|
    KR840006222A|1984-11-22|
    EP0104445A2|1984-04-04|
    YU192183A|1986-12-31|
    PT77380B|1986-03-20|
    ES525876A0|1984-12-01|
    引用文献:
    公开号 | 申请日 | 公开日 | 申请人 | 专利标题
    US4309541A|1978-09-20|1982-01-05|Ciba-Geigy Corporation|Piperidinyl-lactams|
    EP0009465A1|1978-09-20|1980-04-02|Ciba-Geigy Ag|N--3 or 4-piperidyl lactames, process for their preparation and pharmaceutical compositions containing them|
    FR2483920B1|1980-06-09|1983-07-22|Synthelabo|US4601897A|1985-11-06|1986-07-22|Pfizer Inc.|Prazosin-pirbuterol combination for bronchodilation|
    JPS62212385A|1986-03-13|1987-09-18|Kotobuki Seiyaku Kk|Quinazoline derivative and hypotensive agent and production thereof|
    US7799794B2|2000-06-28|2010-09-21|Merck Sharp & Dohme Corp.|Treatment for cardiovascular disease|
    DE60321466D1|2002-07-01|2008-07-17|Tibotec Pharm Ltd|MUTATION PROFILES CORRELATED WITH PHENOTYPIC MEDICAMENT RESISTANCE IN HIV-1 REVERSE TRANSCRIPTASE|
    FR2854633B1|2003-05-07|2005-06-24|Sanofi Synthelabo|PIPERIDINYL-AND PIPERAZINYL-ALKYLCARBAMATES DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE|
    FR2866885B1|2004-02-26|2007-08-31|Sanofi Synthelabo|PIPERIDINYLALKYLCARBAMATES DERIVATIVES, THEIR PREPARATION AND THERAPEUTIC USE THEREOF|
    法律状态:
    优先权:
    申请号 | 申请日 | 专利标题
    DE19823235565|DE3235565A1|1982-09-25|1982-09-25|PIPERIDE DERIVATIVES, THEIR PRODUCTION AND USE|
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